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article · 2015

Metal-free synthesis of 3,5-disubstituted 1H- and 1-aryl-1H-pyrazoles from 1,3-diyne-indole derivatives employing two successive hydroaminations

The uncatalyzed synthesis of 3,5-disubstituted 1<italic>H</italic>- and 1-aryl-1<italic>H</italic>-pyrazoles derived from 1,3-diyne indoles was successfully ...

20 citationsDOI: https://doi.org/10.1039/c4ra16439cOpen accessPDF reported by metadata
Metal-free synthesis of 3,5-disubstituted 1H- and 1-aryl-1H-pyrazoles from 1,3-diyne-indole derivatives employing two successive hydroaminations